CP-809101 hydrochloride
CAS No. 1215721-40-6
CP-809101 hydrochloride ( —— )
产品货号. M26127 CAS No. 1215721-40-6
CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥373 | 有现货 |
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5MG | ¥608 | 有现货 |
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10MG | ¥948 | 有现货 |
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25MG | ¥2090 | 有现货 |
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50MG | ¥3880 | 有现货 |
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100MG | ¥5557 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
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生物学信息
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产品名称CP-809101 hydrochloride
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).
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产品描述CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).(In Vitro):CP-809101 is a potent, functionally selective 5-HT2C agonist that displays approximately 100% efficacy in vitro.(In Vivo):Similar to currently available antipsychotic drugs, CP-809101 dose-dependently inhibited conditioned avoidance responding (CAR, ED50 = 4.8 mg/kg, sc). CP-809101 antagonized both PCP- and d-amphetamine-induced hyperactivity with ED50 values of 2.4 and 2.9 mg/kg (sc), respectively, and also reversed an apomorphine induced-deficit in prepulse inhibition. At doses up to 56 mg/kg, CP-809101 did not produce catalepsy. CP-809101 was inactive in two animal models of antidepressant-like activity, the forced swim test, and learned helplessness.
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同义词——
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体NMDA
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研究领域——
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适应症——
化学信息
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CAS Number1215721-40-6
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分子量341.2
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分子式C15H18Cl2N4O
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纯度>98% (HPLC)
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溶解度——
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SMILESCl.Clc1cccc(COc2cncc(n2)N2CCNCC2)c1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Mikolajczak P et al. Effects of acamprosate and some polyamine site ligands of NMDA receptor on short-term memory in rats. Eur J Pharmacol. 2002 May 24;444(1-2):83-96.
产品手册
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